Affinity DataKi: 0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
Affinity DataKi: 0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0180nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0390nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of DNA-PK in human HeLa nuclear extracts incubated for 40 mins using calf thymus DNA and fluoroscein-p53[Ser15]-peptide by Lanthascreen ti...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Competitive inhibition of Escherichia coli beta-galactosidase assessed as p-nitrophenyl-beta-D-galactopyranoside substrate hydrolysis by UV/Vis spect...More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.346nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nM ΔG°: -12.9kcal/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside substrate measured over 240 mins at 10 mins intervals by U...More data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Arkansas
Curated by PDSP Ki Database
University of Arkansas
Curated by PDSP Ki Database
Affinity DataKi: 1.13nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Competitive inhibition of Escherichia coli beta-galactosidase assessed as p-nitrophenyl-beta-D-galactopyranoside substrate hydrolysis by UV/Vis spect...More data for this Ligand-Target Pair
Affinity DataKi: 1.54nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of bovine liver beta-galactosidase pre-incubated for 30 mins with 4-nitrophenyl-beta-D-galactopyranoside substrate before enzyme addition ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arkansas
Curated by PDSP Ki Database
University of Arkansas
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arkansas
Curated by PDSP Ki Database
University of Arkansas
Curated by PDSP Ki Database
Affinity DataKi: 6.30nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 10.9nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidase using 2-chloro-4-nitrophenyl beta-Dgalactopyranoside as substrate by spectrophotometryMore data for this Ligand-Target Pair